Found 3452 of ki for ALPHA-1B ADRENERGIC RECEPTOR
having polymerids = 3629,7888,11048,49000190,49000199,49000200,49000203 and
complexids = 50002812,50000229,50000717,50006003
having polymerids = 3629,7888,11048,49000190,49000199,49000200,49000203 and
complexids = 50002812,50000229,50000717,50006003
Affinity DataKi: 0.00900nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0380nMAssay Description:Displacement of [3H]prazosin from human recombinant adrenergic alpha-1B receptor expressed in CHO cell membranes incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0390nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.0520nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat cerebral cortex using [3H]prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.0680nMAssay Description:Binding affinity against alpha-1 adrenergic receptor by measuring displacement of [3H]prazosin from rat brain cortex membranes (in vitro).More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Binding affinity against alpha-1 adrenergic receptor by measuring displacement of [3H]prazosin from rat brain cortex membranes (in vitro).More data for this Ligand-Target Pair
Affinity DataKi: 0.0708nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.0810nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0880nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:In vitro binding affinity determined for alpha-1 adrenergic receptor by the displacement of [3H]- prazosin.More data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]prozosin from alpha1b receptor in rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1B adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Binding affinity against alpha-1 adrenergic receptor by measuring displacement of [3H]prazosin from rat brain cortex membranes (in vitro).More data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Binding affinity against Alpha-1B adrenergic receptor from hamster clones.More data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Binding affinity against Alpha-1B adrenergic receptor from hamster clones.More data for this Ligand-Target Pair
Affinity DataKi: 0.129nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.135nMAssay Description:Compound was tested for binding affinity against human hippocampus Alpha-1B adrenergic receptor using radioligand ([3H]-prazosin) binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.135nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.135nMAssay Description:Displacement of [3H]prazosin from Homo sapiens (human) alpha1B adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Binding affinity towards alpha-1 adrenergic receptor from rat brain homogenate preparation by displacement of [3H]prazosinMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Inhibition of [3H]- prazosin binding against Alpha-1B adrenergic receptor from rat liverMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Binding affinity for alpha-1 adrenergic receptor by displacement of [3H]-prazosin from rat brain homogenate preparationMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]prozosin from alpha1b receptor in rat cerebral cortexMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]prozosin from alpha1b receptor in rat cerebral cortexMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Binding affinity for alpha-1 adrenergic receptor by displacement of [3H]-prazosin from rat brain homogenate preparationMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Binding affinity for alpha-1 adrenergic receptor by displacement of [3H]-prazosin from rat brain homogenate preparationMore data for this Ligand-Target Pair
Affinity DataKi: 0.151nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Compound was tested for the inhibition of [3H]prazosin binding Alpha-1 adrenergic receptor of crude rat brain membrane.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Binding affinity towards alpha-1 adrenergic receptor from rat brain homogenate preparation by displacement of [3H]prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Binding affinity to Alpha-1 adrenergic receptor by displacement of [3H]prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Binding affinity against alpha-1 adrenergic receptor by measuring displacement of [3H]prazosin from rat brain cortex membranes (in vitro).More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:In vitro binding affinity determined for alpha-1 adrenergic receptor by the displacement of [3H]- prazosin.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Binding affinity against alpha-1-adrenoceptor was determined by displacement of [3H]-prazosin in rat brain homogenates.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:In vitro binding affinity towards Alpha-1 adrenergic receptor was determined by the displacement of [3H]prazosinMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Compound was tested for its binding affinity for alpha-1 adrenergic receptor site by displacement of [3H]clonidine at 10e-6 M concentrationMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.191nMAssay Description:Displacement of [3H]prazosin from human alpha1B adrenergic receptor expressed in CHO cell membranes after 30 mins by rapid filtration methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:In vitro binding affinity determined for alpha-1 adrenergic receptor by the displacement of [3H]- prazosin.More data for this Ligand-Target Pair